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GSK-25
GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K (RSK1 IC50 of 398 nM, p70S6K IC50 of 1000nM), and a dramatically improved P450 profile (>2.2 uM at all isozymes tested).
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GSK-25
GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K (RSK1 IC50 of 398 nM, p70S6K IC50 of 1000nM), and a dramatically improved P450 profile (>2.2 uM at all isozymes tested).
TargetMol | 1 mg | ￥9,000 | ||
| 2 mg | ￥12,500 | ||
| 5 mg | ￥19,500 | ||
| 10 mg | ￥27,500 | ||
| 25 mg | ￥41,500 | ||
| 50 mg | ￥66,000 | ||
| 100 mg | ￥110,000 | ||
| 1 mL x 10 mM (in DMSO) | ￥22,000 |
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関連 阻害 剤 製品 "GSK-25"
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製品 情報
GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K (RSK1 IC50 of 398 nM, p70S6K IC50 of 1000nM), and a dramatically improved P450 profile (>2.2 uM at all isozymes tested). | |
| Targets&IC50 | mTOR (p70S6K):1000nM, RSK1:398 nM |
| Alias | GSK25 |
| 513.33 | |
| C24H16Cl2F2N6O | |
| CAS | 874119-56-9 |
| Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||||||||||||||||||
DMSO: 60 mg/mL (116.88 mM)  | ||||||||||||||||||||||||||||||||||||
DMSO
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計算 機
投与 溶液 組成 計算 （完全 溶解 ）
となります。10
DMSO+30% PEG300+5% Tween 80+60% ddH2O. という , 300 を を600用量 換算
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Keywords
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Related Tags: buy GSK-25 | purchase GSK-25 | GSK-25 cost | order GSK-25 | GSK-25 chemical structure | GSK-25 formula | GSK-25 molecular weight
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