别孕烷醇酮
Zulresso | |
其他 | ALLO; Allo; ALLOP; AlloP; Brexanolone; SAGE-547; SGE-102; 5 |
给药 | Intravenous infusion[1] |
Neurosteroids; Antidepressants | |
>99%[1] | |
药物 | Non-CYP450 (keto-reduction via AKRs, glucuronidation via UGTs, sulfation via SULTs)[1] |
9 hours[1] | |
Feces: 47%[1] Urine: 42%[1] | |
识别 | |
| |
CAS | 516-54-1 |
PubChem CID | |
DrugBank | |
ChemSpider | |
UNII | |
KEGG | |
ChEBI | |
ChEMBL | |
CompTox Dashboard (EPA) | |
C21H34O2 | |
318.501 g/mol | |
3D | |
| |
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别孕烷醇酮(
参考 文献
[编辑]- ^ 1.0 1.1 1.2 1.3 1.4 1.5
存 档副本 (PDF). [2019-05-26]. (原始 内容 存 档 (PDF)于2020-11-12). - ^ Reddy DS. Neurosteroids: endogenous role in the human brain and therapeutic potentials. Progress in Brain Research 186. 2010: 113–37. ISBN 9780444536303. PMC 3139029 . PMID 21094889. doi:10.1016/B978-0-444-53630-3.00008-7.
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被 忽 略 (帮助) - ^ 3.0 3.1 Commissioner, Office of the. Press Announcements - FDA approves first treatment for post-partum depression. www.fda.gov. [21 March 2019]. (
原始 内容 存 档于2019-04-22) (英 语). - ^ Frieder A, Fersh M, Hainline R, Deligiannidis KM. Pharmacotherapy of Postpartum Depression: Current Approaches and Novel Drug Development. CNS Drugs. March 2019, 33 (3): 265–282. PMID 30790145. doi:10.1007/s40263-019-00605-7.
- ^ Wilkinson ST, Sanacora G. A new generation of antidepressants: an update on the pharmaceutical pipeline for novel and rapid-acting therapeutics in mood disorders based on glutamate/GABA neurotransmitter systems. Drug Discov. Today. February 2019, 24 (2): 606–615. PMID 30447328. doi:10.1016/j.drudis.2018.11.007.